SCHEMBL6300285

SCHEMBL6300285

Nc1ccc(-n2nnn(CCCOc3ccc(F)cc3)c2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
CYP2C19 P33261 1/20 0.41
MAOB P27338 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HTR1A P08908 3/20 0.39
DRD2 P14416 3/20 0.39
HTR2A P28223 3/20 0.39
DRD3 P35462 3/20 0.39
DRD1 P21728 2/20 0.39
POLB P06746 1/20 0.39
DRD5 P21918 1/20 0.39
RAB9A P51151 2/20 0.39
ATM Q13315 1/20 0.39
SIGMAR1 Q99720 2/20 0.38
HRH1 P35367 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
KCNH2 Q12809 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
PLA2G7 Q13093 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6300283 0.86 PARP10 (0.47) NPC1CYP2C19MAOBHRH1KCNH2
SCHEMBL4673533 0.84 ENPP2 (0.44) DRD2DRD3POLBHRH3
SCHEMBL4672126 0.75 NPBWR1 (0.42) DRD2SIGMAR1
SCHEMBL4670427 0.73 ADORA2B (0.41)
SCHEMBL4670482 0.73 DHODH (0.36) NPC1CYP2C19MAOBRXFP1RAB9A
SCHEMBL4673358 0.72 MAOB (0.46) MAOBSIGMAR1
Hydrochloric Acid SCHEMBL9384727 0.72 ADORA2B (0.40)
SCHEMBL6301320 0.71 ADRB2 (0.41)
Water SCHEMBL4673070 0.70 ADRB2 (0.42)
Water SCHEMBL4672111 0.70 ADRB2 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6903218-B2 Sulfonamide substituted chroman derivatives BAYER PHARMACEUTICALS CORPORATION (US) 2005-06-07 US disclosed