SCHEMBL4687459

SCHEMBL4687459

Nc1c(Cl)cc(F)cc1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.43
CSNK2A1 P68400 2/20 0.41
METAP2 P50579 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 1/20 0.39
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
GLA P06280 1/20 0.38
ACLY P53396 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
HTT P42858 1/20 0.37
MAP4K4 O95819 1/20 0.37
GRM2 Q14416 1/20 0.36
SMARCA2 P51531 1/20 0.36
SMARCA4 P51532 1/20 0.36
PBRM1 Q86U86 1/20 0.36
P2RX7 Q99572 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28871472 0.86 PTGS2 (0.42) ALDH1A1SMN1; SMN2KDM4EMEN1KMT2A
SCHEMBL22616582 0.85 TAAR1 (0.47) ALDH1A1KDM4EMEN1KMT2AMAP4K4
SCHEMBL4787759 0.85 AHR (0.42) HSD17B10SMN1; SMN2MEN1KMT2AMAP4K4
SCHEMBL3651531 0.81 PLA2G7 (0.44) CYP2A6ALDH1A1HSD17B10HPGDSMN1; SMN2
SCHEMBL30579808 0.80 CYP2A6 (0.46) CYP2A6CSNK2A1METAP2ALDH1A1HPGD
SCHEMBL7246163 0.80 CYP2A6 (0.46) CYP2A6CSNK2A1ALDH1A1HSD17B10HPGD
SCHEMBL5174258 0.80 ALDH1A1 (0.52) CYP2A6CSNK2A1ALDH1A1HSD17B10HPGD
SCHEMBL28106449 0.80 METAP2 (0.42) METAP2ALDH1A1HSD17B10HPGDSMARCA2
SCHEMBL19857180 0.77 METAP2 (0.40) CYP2A6METAP2ALDH1A1HSD17B10HPGD
SCHEMBL29972900 0.76 GRM2 (0.42) CYP2A6CSNK2A1MAP4K4GRM2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114072393-B 3-Amino-4H-benzo [ E ] [1,2,4] thiadiazine 1, 1-dioxide derivatives as MRGX2 inhibitors 索伦特治疗有限责任公司 2025-05-27 CN disclosed
EP-1965642-A2 PYRAZOLYL CARBOXAMIDES Bayer CropScience AG (DE) 2008-09-10 EP disclosed
WO-2007068370-A2 PYRAZOLYL CARBOXAMIDES BAYER CROPSCIENCE AG (DE) 2007-06-21 WO disclosed