SCHEMBL4688387

SCHEMBL4688387

CCCC(=O)OC(=O)c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.51
ALDH1A1 P00352 4/20 0.48
KMT2A Q03164 5/20 0.46
MEN1 O00255 4/20 0.46
MAPT P10636 2/20 0.46
CASP3 P42574 1/20 0.46
TRPV1 Q8NER1 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
MAPK1 P28482 2/20 0.44
HTT P42858 1/20 0.44
ATM Q13315 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 2/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
HPGD P15428 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20485512 0.91 ALDH1A1 (0.58) ALDH1A1KMT2AMAPTNPC1RAB9A
SCHEMBL27200589 0.90 HTR7 (0.62) HTR7KMT2AMEN1MAPTCASP3
SCHEMBL5560398 0.87 KMT2A (0.50) HTR7ALDH1A1KMT2AMEN1MAPT
SCHEMBL7164306 0.87 GAA (0.55) HTR7ALDH1A1KMT2AMEN1MAPT
SCHEMBL10579985 0.84 HSD17B3 (0.58) ALDH1A1KMT2AMEN1MAPTMAPK1
SCHEMBL8995839 0.84 TDP1 (0.52) ALDH1A1KMT2AMAPTTRPV1NPC1
SCHEMBL8591084 0.82 ALDH1A1 (0.48) ALDH1A1KMT2AMEN1MAPTNPC1
SCHEMBL8995791 0.82 ALDH1A1 (0.48) ALDH1A1KMT2AMEN1MAPTNPC1
Hydrogen Peroxide SCHEMBL29219018 0.81 LMNA (0.56) ALDH1A1KMT2AMAPK1CES2CES1
SCHEMBL266279 0.81 LMNA (0.56) ALDH1A1KMT2AMAPK1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103694111-B A kind of preparation method of 4-(4-fluoro benzoyl) butyric acid ZHEJIANG XINHECHENG CO., LTD. (CN) 2016-02-03 CN claimed
CN-103694111-A Method for preparing 4-(4-fluorobenzoyl) butyric acid ZHEJIANG NHU CO LTD 2014-04-02 CN claimed
EP-2004639-A2 PROCESSES FOR THE SYNTHESIS OF AZETIDINONE Teva Pharmaceutical Industries Ltd (IL) 2008-12-24 EP claimed
US-20080032964-A1 Process for the synthesis of azetidinone TEVA PHARMACEUTICALS USA, INC. 2008-02-07 US claimed
WO-2007120824-A2 PROCESSES FOR THE SYNTHESIS OF AZETIDINONE TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2007-10-25 WO claimed
CN-116981655-A Haizimabu intermediate and preparation method thereof 浙江海正药业股份有限公司 2023-10-31 CN disclosed
CN-109942523-B Benzofuran and benzofuran coumarin derivatives, and preparation method and application thereof 华东师范大学 2023-06-09 CN disclosed
CN-115583962-A Isomer of ezetimibe key intermediate and preparation method thereof 山东新时代药业有限公司 2023-01-10 CN disclosed
CN-115184485-A Ezetimibe prodrug impurity detection method 南京优科生物医药股份有限公司 2022-10-14 CN disclosed
CN-114989123-A Flavone-3-carboxylic acid compound, bactericidal composition containing compound and application 长江大学 2022-09-02 CN disclosed
CN-107488164-A A kind of Ezetimibe intermediate compound 山东新时代药业有限公司 2017-12-19 CN disclosed
CN-107488173-A A kind of Ezetimibe intermediate and its synthetic method 山东新时代药业有限公司 2017-12-19 CN disclosed
US-5145959-A Enzyme inhibitors; antilipemic agents; treatment of atherosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1992-09-08 US disclosed
US-5075311-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1991-12-24 US disclosed
EP-0356788-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1990-03-07 EP disclosed
US-4517301-A URINALYSIS, METAL SALT OF BETA-KETO ACID/ESTER MILES LABORATORIES, INC. (US) 1985-05-14 US disclosed
EP-0051209-B1 DEVICE AND METHOD FOR PREPARATION OF A CONTROL SOLUTION FOR KETONE DETERMINATION MILES LABORATORIES, INC. (US) 1985-01-16 EP disclosed
EP-0029915-B1 DEVICE AND METHOD FOR THE PREPARATION OF A CONTROL SOLUTION FOR KETONE DETERMINATION AND METHOD OF CALIBRATING A KETONE TEST INSTRUMENT MILES LABORATORIES, INC. (US) 1983-07-20 EP disclosed
EP-0051209-A1 Device and method for preparation of a control solution for ketone determination MILES LABORATORIES, INC. (US) 1982-05-12 EP disclosed
EP-0029915-A1 Device and method for the preparation of a control solution for ketone determination and method of calibrating a ketone test instrument MILES LABORATORIES, INC. (US) 1981-06-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080032964-A1 Process for the synthesis of azetidinone CYP46A1, APOB, CYP51A1 HTR7 1119/4885ALDH1A1 464/4885KMT2A 1017/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.