SCHEMBL4690185

SCHEMBL4690185

CC(CN1C[C@@H](C(=O)N2CC3CN(CC[CH]c4ccccc4)CC3C2)CC1=O)C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.38
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
CCR5 P51681 2/20 0.34
CCL5 P13501 1/20 0.34
KMT2A Q03164 2/20 0.33
PKM P14618 1/20 0.33
NPC1 O15118 1/20 0.33
P2RX7 Q99572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694943 0.82 NPC1 (0.34) ALDH1A1MAPK1HTTCCR5CCL5
SCHEMBL4695010 0.78 KMT2A (0.38) POLBALDH1A1CCR5CCL5KMT2A
SCHEMBL4690190 0.76 POLB (0.49) POLBALDH1A1CYP1A2MAPK1HTT
SCHEMBL4692061 0.76 CCR5 (0.37) ALDH1A1CYP1A2CCR5CCL5
SCHEMBL4695866 0.74 CCR5 (0.36) ALDH1A1CCR5CCL5KMT2A
SCHEMBL4694234 0.74 ALDH1A1 (0.41) ALDH1A1MAPK1HTTNPC1
SCHEMBL4696881 0.73 CCL5 (0.38) ALDH1A1CCR5CCL5
SCHEMBL4692848 0.73 ALDH1A1 (0.40) POLBALDH1A1CCR5CCL5KMT2A
SCHEMBL4692781 0.72 PKM (0.36) ALDH1A1CYP1A2MAPK1CCR5CCL5
SCHEMBL4695377 0.71 CCR5 (0.37) CYP1A2CCR5CCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed