SCHEMBL4690443

SCHEMBL4690443

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)[C@@H]3CN(Cc4ccccc4)CCO3)CC2C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.37
DRD4 P21917 6/20 0.36
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
CYP2C19 P33261 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
FAAH O00519 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
GRN P28799 1/20 0.34
SORT1 Q99523 1/20 0.34
JAK2 O60674 2/20 0.34
JAK3 P52333 2/20 0.34
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
BCHE P06276 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694985 0.84 GRIN2B (0.44) GRIN2BDRD2DRD3
SCHEMBL3282844 0.84 GRIN2B (0.44) GRIN2BDRD2DRD3
SCHEMBL4694234 0.80 ALDH1A1 (0.41) ALDH1A1
SCHEMBL4690448 0.79 GRIN2B (0.41) GRIN2BDRD4DRD2DRD3CYP2C19
SCHEMBL4693059 0.78 CCR5 (0.37) KDM4EALDH1A1
SCHEMBL4693208 0.76 CCR5 (0.42)
SCHEMBL4692078 0.76 CCR5 (0.40)
SCHEMBL4694455 0.76 CHRNB2 (0.44) ALDH1A1HPGD
SCHEMBL4693659 0.76 CHRNB2 (0.47) KDM4EALDH1A1
SCHEMBL4694380 0.76 FAAH (0.41) DRD4DRD2KDM4EALDH1A1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed