SCHEMBL4690155

SCHEMBL4690155

NC(=O)n1ccc(C(=O)N2CC3CN(CC[CH]c4ccccc4)C[C@H]3C2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
FAAH O00519 4/20 0.35
MGLL Q99685 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CCR5 P51681 6/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 2/20 0.34
HSD17B10 Q99714 2/20 0.34
USP2 O75604 1/20 0.34
CCL5 P13501 4/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNB4 P30926 2/20 0.33
CHRNA3 P32297 2/20 0.33
CHRNA7 P36544 2/20 0.33
CHRNA4 P43681 2/20 0.33
F2 P00734 1/20 0.33
PLAU P00749 1/20 0.33
KLKB1 P03952 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694094 0.79 CHRNB2 (0.44) HPGDSMN1; SMN2CCR5ALDH1A1CHRNB2
SCHEMBL4694116 0.78 HCRTR2 (0.38) CCR5CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4690538 0.78 CCL5 (0.36) CCR5CCL5
SCHEMBL4694680 0.78 ALK (0.34) MEN1KMT2ACCR5CCL5CHRNB2
SCHEMBL4692781 0.77 PKM (0.36) MEN1HPGDKMT2ACCR5ALDH1A1
SCHEMBL4690761 0.76 KDM4E (0.43) MEN1HPGDKMT2ASMN1; SMN2CCR5
SCHEMBL4695377 0.76 CCR5 (0.37) CCR5TSHRHSD17B10CCL5CHRNB2
SCHEMBL4692820 0.75 CCL5 (0.35) CCR5ALDH1A1CCL5KDM4EHTT
SCHEMBL4690459 0.75 MEN1 (0.37) MEN1KMT2ACCR5ALDH1A1CCL5
SCHEMBL4693281 0.75 CHRNB2 (0.43) MEN1KMT2ASMN1; SMN2CCR5TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed