SCHEMBL4690840

SCHEMBL4690840

Cc1ccc(NC(=O)CCN2CC3CN(C(=O)c4ccc(C(F)(F)F)cc4)CC3C2)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY2R P49146 1/20 0.49
RXFP1 Q9HBX9 1/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C19 P33261 3/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 1/20 0.47
UBE2M P61081 1/20 0.46
DCUN1D1 Q96GG9 1/20 0.46
CYP2D6 P10635 2/20 0.46
EPHX2 P34913 1/20 0.45
PRKAB2 O43741 3/20 0.44
PRKAG1 P54619 3/20 0.44
PRKAA2 P54646 3/20 0.44
PRKAA1 Q13131 3/20 0.44
PRKAG3 Q9UGI9 3/20 0.44
PRKAG2 Q9UGJ0 3/20 0.44
PRKAB1 Q9Y478 3/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 2/20 0.43
MEN1 O00255 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694150 0.90 NPY2R (0.51) NPY2RRXFP1CYP3A4CYP2C19CYP1A2
SCHEMBL4695754 0.90 CYP1A2 (0.46) RXFP1CYP3A4CYP2C19CYP1A2CYP2C9
SCHEMBL4695971 0.89 LMNA (0.50) CYP3A4CYP2C19CYP1A2CYP2C9UBE2M
SCHEMBL4691227 0.88 CYP1A2 (0.46) RXFP1CYP3A4CYP2C19CYP1A2CYP2C9
SCHEMBL4691875 0.88 CYP3A4 (0.46) RXFP1CYP3A4CYP2C19CYP1A2CYP2C9
SCHEMBL4690531 0.86 MAPT (0.48) CYP3A4CYP2C19CYP1A2CYP2C9UBE2M
SCHEMBL4692068 0.86 ALDH1A1 (0.49) CYP3A4CYP2C19CYP1A2CYP2C9UBE2M
SCHEMBL4690845 0.86 NPY2R (0.46) NPY2RRXFP1UBE2MDCUN1D1EPHX2
SCHEMBL4689516 0.86 MAPT (0.61) TP53MAPTKMT2ALMNAPOLB
SCHEMBL4693588 0.85 UBE2M (0.46) CYP3A4CYP2C19CYP1A2CYP2C9UBE2M

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed