SCHEMBL4692204

SCHEMBL4692204

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4c(C)sc(C)c4C#N)CC3C2)cc1Cl

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
KDM1A O60341 1/20 0.33
TNF P01375 1/20 0.33
CCR5 P51681 6/20 0.32
CCL5 P13501 1/20 0.32
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
FASN P49327 2/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695956 0.89 HCRTR1 (0.37) HCRTR1HCRTR2TNFCCR5
SCHEMBL4693134 0.87 HCRTR1 (0.36) HCRTR1HCRTR2TNFCCR5
SCHEMBL4695625 0.87 HCRTR1 (0.34) HCRTR1HCRTR2KDM1ATNFCCR5
SCHEMBL4694334 0.83 HCRTR1 (0.43) HCRTR1HCRTR2TNFCCR5CCL5
SCHEMBL4690403 0.83 HCRTR1 (0.39) HCRTR1HCRTR2TNFCCR5
SCHEMBL3281863 0.83 HCRTR1 (0.48) HCRTR1HCRTR2TNFCCR5
SCHEMBL4693590 0.82 KDM1A (0.48) KDM1AFASN
SCHEMBL4692864 0.81 TNF (0.35) HCRTR1HCRTR2TNFCCR5GAA
SCHEMBL4693907 0.81 HCRTR1 (0.48) HCRTR1HCRTR2KDM1ATNFCCR5
SCHEMBL4694248 0.81 ALDH1A1 (0.39) HCRTR1HCRTR2TNFCCR5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed