SCHEMBL4694248

SCHEMBL4694248

Cc1ccc(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)s1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
TNF P01375 1/20 0.36
EPHX2 P34913 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
HCRTR1 O43613 2/20 0.33
HCRTR2 O43614 2/20 0.33
CCR5 P51681 1/20 0.33
TACR2 P21452 1/20 0.32
TACR1 P25103 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
S1PR1 P21453 1/20 0.31
HRH4 Q9H3N8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692864 0.86 TNF (0.35) ALDH1A1HPGDTNFGAAHCRTR1
SCHEMBL4695956 0.84 HCRTR1 (0.37) HPGDTNFHCRTR1HCRTR2CCR5
SCHEMBL4690403 0.83 HCRTR1 (0.39) ALDH1A1HPGDTNFHCRTR1HCRTR2
SCHEMBL4694334 0.83 HCRTR1 (0.43) TNFEPHX2HCRTR1HCRTR2CCR5
SCHEMBL3281863 0.83 HCRTR1 (0.48) TNFHCRTR1HCRTR2CCR5
SCHEMBL4694340 0.83 TNF (0.36) ALDH1A1TNFLMNAHCRTR1HCRTR2
SCHEMBL4692886 0.83 ALDH1A1 (0.42) ALDH1A1HPGDTNFHCRTR1HCRTR2
SCHEMBL4695935 0.83 HCRTR2 (0.47) ALDH1A1HPGDTNFHCRTR1HCRTR2
SCHEMBL4695972 0.83 CHRNB2 (0.40) ALDH1A1HPGDTNFGAAHCRTR1
SCHEMBL4693134 0.83 HCRTR1 (0.36) TNFHCRTR1HCRTR2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed