SCHEMBL4693590

SCHEMBL4693590

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4ccc(C#N)cc4)CC3C2)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.48
ALDH1A1 P00352 1/20 0.43
FASN P49327 17/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691612 0.87 KDM1A (0.38) KDM1AALDH1A1FASN
SCHEMBL4695972 0.87 CHRNB2 (0.40) ALDH1A1
SCHEMBL4692070 0.86 HPGD (0.36) KDM1AALDH1A1
SCHEMBL4689519 0.86 ALDH1A1 (0.47) ALDH1A1
SCHEMBL4690534 0.85 LMNA (0.39)
SCHEMBL4690843 0.85 GAA (0.41)
SCHEMBL4695193 0.85 TRPV4 (0.40) KDM1A
SCHEMBL4693907 0.84 HCRTR1 (0.48) KDM1A
SCHEMBL4694328 0.83 TNF (0.35) KDM1AALDH1A1
SCHEMBL4691641 0.83 CHRNB2 (0.43) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed