SCHEMBL4692864

SCHEMBL4692864

Cc1cc(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)c(C)s1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.35
HCRTR1 O43613 7/20 0.35
HCRTR2 O43614 7/20 0.35
USP2 O75604 1/20 0.32
GAA P10253 1/20 0.32
PKM P14618 1/20 0.32
TSHR P16473 1/20 0.32
CCR5 P51681 1/20 0.31
HPGD P15428 2/20 0.31
ALDH1A1 P00352 1/20 0.31
MGLL Q99685 1/20 0.31
HTR1A P08908 1/20 0.31
S1PR1 P21453 1/20 0.30
HRH4 Q9H3N8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694248 0.86 ALDH1A1 (0.39) TNFHCRTR1HCRTR2GAACCR5
SCHEMBL4695935 0.86 HCRTR2 (0.47) TNFHCRTR1HCRTR2HPGDALDH1A1
SCHEMBL4692886 0.86 ALDH1A1 (0.42) TNFHCRTR1HCRTR2CCR5HPGD
SCHEMBL4695956 0.85 HCRTR1 (0.37) TNFHCRTR1HCRTR2CCR5HPGD
SCHEMBL4690680 0.85 HCRTR1 (0.42) TNFHCRTR1HCRTR2HPGDALDH1A1
SCHEMBL4690738 0.85 HCRTR1 (0.46) TNFHCRTR1HCRTR2HPGDALDH1A1
SCHEMBL4692692 0.85 HCRTR1 (0.45) TNFHCRTR1HCRTR2TSHRALDH1A1
SCHEMBL4694354 0.84 P2RX7 (0.44) TNFHCRTR1HCRTR2
SCHEMBL4691868 0.84 HCRTR1 (0.47) TNFHCRTR1HCRTR2CCR5ALDH1A1
SCHEMBL4693718 0.84 TSHR (0.38) TNFHCRTR1HCRTR2TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed