Nitric Acid

Nitric Acid

SCHEMBL4693602

CC(C)(C)[Si](O[Si](c1ccccc1)(c1ccccc1)C(C)(C)C)(c1ccccc1)c1ccccc1.O=[N+]([O-])O.O=[N+]([O-])O.O=[N+]([O-])O.OCC(CO)(CO)CO

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ERG11

The experimentally established mechanism targets of Nitric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.37
GSR P00390 1/20 0.33
ALDH1A1 P00352 4/20 0.33
HTT P42858 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 2/20 0.32
SMYD2 Q9NRG4 2/20 0.31
HSP90AA1 P07900 1/20 0.31
LTB4R Q15722 1/20 0.31
NPSR1 Q6W5P4 2/20 0.31
MAPT P10636 4/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
F2R P25116 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
F2RL3 Q96RI0 1/20 0.30
NPBWR1 P48145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7597173 0.89 MGAM (0.35) ABL1ALDH1A1HTTSMYD2NPSR1
SCHEMBL79874 0.78 MAPK1 (0.37) ALDH1A1HTTSMYD2SMN1; SMN2
Nitric Acid SCHEMBL3869559 0.77 LTB4R (0.32) ABL1ALDH1A1HTTSMYD2LTB4R
Hydroxyamine SCHEMBL9901947 0.76 ALDH1A1 (0.35) ALDH1A1SMYD2MAPTKMT2A
SCHEMBL2955809 0.74 SMYD2 (0.33) HTTSMYD2NPSR1KDM4ESMN1; SMN2
SCHEMBL8027742 0.74 SMYD2 (0.33) HTTSMYD2NPSR1KDM4ESMN1; SMN2
1,3-Butanediol SCHEMBL3804833 0.74 TRPA1 (0.36) LMNASMYD2
SCHEMBL4693599 0.71 ALDH1A1 (0.46) ABL1ALDH1A1HTTLMNASMYD2
SCHEMBL28978518 0.70 NPSR1 (0.33) ALDH1A1HTTSMYD2NPSR1SMN1; SMN2
SCHEMBL3869948 0.70 SMYD2 (0.35) HTTSMYD2LTB4RSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109542-A4 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-03-26 EP disclosed
US-6469065-B1 COMPOUND THAT DONATES, TRANSFERS OR RELEASES NITRIC OXIDE, ELEVATES ENDOGENOUS LEVELS OF NITRIC OXIDE NITROMED, INC. 2002-10-22 US disclosed
US-20020143007-A1 Nitrosated and nitrosylated alpha-adrenergic receptor antagonists, compositions and methods of use GARVEY DAVID S (US) 2002-10-03 US disclosed
EP-1109542-A1 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2001-06-27 EP disclosed
WO-2000012075-A1 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2000-03-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020143007-A1 Nitrosated and nitrosylated alpha-adrenergic receptor antagonists, compositions and methods of use ADRB1, ADRB3, ADRA1D ABL1 3711/4885GSR 389/4885ALDH1A1 610/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.