SCHEMBL4693889

SCHEMBL4693889

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4nccc5ccccc45)CC3C2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 2/20 0.44
HCRTR1 O43613 11/20 0.41
HCRTR2 O43614 10/20 0.41
PDE2A O00408 1/20 0.40
CHRM2 P08172 1/20 0.39
EPHX2 P34913 1/20 0.36
TNF P01375 1/20 0.36
PDE4B Q07343 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689931 0.87 HCRTR1 (0.39) HCRTR1HCRTR2TNFPDE4B
SCHEMBL4693290 0.87 PDE10A (0.40) HCRTR1HCRTR2PDE2AEPHX2TNF
SCHEMBL4691532 0.84 CHRNB2 (0.44) HCRTR1HCRTR2TNFPDE4B
SCHEMBL3282223 0.82 CCR5 (0.43) HCRTR1HCRTR2CHRM2
SCHEMBL4693800 0.81 RAB9A (0.43) HCRTR1HCRTR2PDE2ATNF
SCHEMBL4695972 0.81 CHRNB2 (0.40) HCRTR1HCRTR2TNF
SCHEMBL4692886 0.81 ALDH1A1 (0.42) HCRTR1HCRTR2TNF
SCHEMBL4690542 0.81 HCRTR1 (0.39) HCRTR1HCRTR2PDE2ATNFPDE4B
SCHEMBL4694845 0.81 HCRTR1 (0.37) HCRTR1HCRTR2TNF
SCHEMBL3281863 0.80 HCRTR1 (0.48) HCRTR1HCRTR2TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed