SCHEMBL4694474

SCHEMBL4694474

NC(=O)C1[C@@H]2CN(C(=O)c3cccc(F)c3)CC2CN1CC[CH]c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.40
USP2 O75604 2/20 0.39
GRM5 P41594 2/20 0.39
PLA2G7 Q13093 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
NPY5R Q15761 1/20 0.38
CYP2D6 P10635 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
KMT2A Q03164 1/20 0.37
CHRNB2 P17787 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5232784 0.91 CHRNB2 (0.43) SMN1; SMN2ALDH1A1HPGDMEN1KMT2A
SCHEMBL5236245 0.86 GRM5 (0.42) GRM5ALDH1A1CYP3A4CHRNB2CHRNB4
SCHEMBL4694489 0.86 HCRTR1 (0.35) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL4692727 0.84 SIGMAR1 (0.40) KMT2A
SCHEMBL3283159 0.83 CHRNB2 (0.47) MAPK1SMN1; SMN2NPY5RALDH1A1HPGD
SCHEMBL4691561 0.82 CHRM2 (0.36) SMN1; SMN2NPY5RALDH1A1MEN1KMT2A
SCHEMBL5236634 0.82 ALDH1A1 (0.42) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL5235762 0.82 CHRNB2 (0.44) SMN1; SMN2ALDH1A1HPGDMEN1KMT2A
SCHEMBL5235903 0.82 CCR5 (0.40) SMN1; SMN2HPGDMEN1KMT2ACHRNB2
SCHEMBL4694358 0.81 DPP4 (0.45) SMN1; SMN2ALDH1A1HPGDCYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed