SCHEMBL5236245

SCHEMBL5236245

N#Cc1cccc(C(=O)N2CC3CN(CC[CH]c4ccccc4)C(C(N)=O)[C@@H]3C2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.42
ALDH1A1 P00352 2/20 0.37
KCNA5 P22460 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
SLC9A1 P19634 1/20 0.35
CYP2C19 P33261 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
GRIN2B Q13224 2/20 0.35
SMO Q99835 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
BACE1 P56817 1/20 0.34
NAMPT P43490 2/20 0.34
MGLL Q99685 1/20 0.34
GSK3B P49841 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236634 0.91 ALDH1A1 (0.42) ALDH1A1KCNA5CHRNB2CHRNB4CHRNA3
SCHEMBL5232784 0.89 CHRNB2 (0.43) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4694474 0.86 MAPK1 (0.40) GRM5ALDH1A1CYP3A4CHRNB2CHRNB4
SCHEMBL3283159 0.81 CHRNB2 (0.47) ALDH1A1CYP3A4CYP2C9CHRNB2CHRNB4
SCHEMBL5235762 0.80 CHRNB2 (0.44) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4691561 0.80 CHRM2 (0.36) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL5235903 0.80 CCR5 (0.40) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL5235498 0.79 HDAC3 (0.38) ALDH1A1CYP3A4CHRNB2CHRNB4CHRNA3
SCHEMBL4694358 0.79 DPP4 (0.45) ALDH1A1CYP3A4MGLL
SCHEMBL4689727 0.78 DPP4 (0.45) CHRNB2CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed