SCHEMBL4697059

SCHEMBL4697059

O=C(O)C1c2nn(C(c3ccccc3)(c3ccccc3)c3ccccc3)cc2C(NOCc2ccccc2)CN1C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 1/20 0.32
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC11 Q96DB2 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
HDAC9 Q9UKV0 1/20 0.30
HDAC5 Q9UQL6 1/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4130806 0.92 GPR183 (0.32) AGTR2HDAC3HDAC4HDAC1HDAC7
SCHEMBL20558122 0.83 GHSR (0.36) AGTR2
SCHEMBL4695538 0.79
SCHEMBL5254943 0.78 NPC1 (0.38) NPC1RAB9AEPHX2
SCHEMBL4147803 0.73 MMP2 (0.32)
SCHEMBL4697074 0.72 NPC1 (0.34) AGTR2NPC1RAB9AEPHX2
SCHEMBL3305431 0.72 LMNA (0.34) NPC1RAB9AEPHX2
SCHEMBL4695600 0.71 KEAP1 (0.40) NPC1RAB9A
SCHEMBL5187275 0.71 GPR183 (0.39) NPC1RAB9A
SCHEMBL20557469 0.70 MEN1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed