SCHEMBL4699471

SCHEMBL4699471

CC(C)C[C@@H](C(N)=O)N(CC#N)c1cscc1-c1ccc(CNCC(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.36
GRM2 Q14416 1/20 0.36
CTSS P25774 6/20 0.34
CTSK P43235 5/20 0.34
CTSL P07711 5/20 0.34
CTSB P07858 5/20 0.34
PRKD1 Q15139 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701072 0.88 PDCD1 (0.35) CTSSCTSKCTSLCTSB
SCHEMBL4704896 0.88 CTSK (0.34) CTSSCTSKCTSLCTSB
SCHEMBL4703639 0.86 CTSK (0.36) CTSSCTSKCTSLCTSBPRKD1
SCHEMBL4699572 0.86 CTSL (0.33) CTSSCTSKCTSLCTSB
SCHEMBL4704688 0.82 CTSL (0.33) CTSSCTSKCTSLCTSB
SCHEMBL4703317 0.82 HRH3 (0.35) CTSSCTSKCTSLCTSB
SCHEMBL4703612 0.81 CTSS (0.34) CTSSCTSKCTSLCTSB
SCHEMBL4703463 0.81 HRH3 (0.37) KCNH2CTSSCTSKCTSLCTSB
SCHEMBL4701830 0.81 CTSK (0.37) CTSSCTSKCTSLCTSB
SCHEMBL4699887 0.80 CTSS (0.34) CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed