SCHEMBL4703463

SCHEMBL4703463

CC(C)C[C@@H](C(N)=O)N(CC#N)c1cscc1-c1ccc(CNCCCN2CCCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.37
HRH1 P35367 1/20 0.37
HDAC1 Q13547 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
KMT2A Q03164 2/20 0.33
OPRK1 P41145 5/20 0.33
OPRM1 P35372 4/20 0.33
HTR3A P46098 2/20 0.33
OPRD1 P41143 1/20 0.32
KCNH2 Q12809 1/20 0.32
PDGFRB P09619 1/20 0.32
KDR P35968 1/20 0.32
SLC2A1 P11166 2/20 0.32
MEN1 O00255 1/20 0.32
RAD52 P43351 1/20 0.32
ATM Q13315 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701072 0.87 PDCD1 (0.35) CTSLCTSBCTSSCTSK
SCHEMBL4703746 0.86 OPRM1 (0.37) HRH3CTSLCTSBCTSSCTSK
SCHEMBL4703639 0.83 CTSK (0.36) CTSLCTSBCTSSCTSK
SCHEMBL4704896 0.83 CTSK (0.34) CTSLCTSBCTSSCTSK
SCHEMBL4699572 0.83 CTSL (0.33) HDAC1CTSLCTSBCTSSCTSK
SCHEMBL4699471 0.81 KCNH2 (0.36) CTSLCTSBCTSSCTSKKCNH2
SCHEMBL4701956 0.78 SPHK1 (0.39) HRH3CTSLCTSBCTSSCTSK
SCHEMBL4704688 0.78 CTSL (0.33) HRH3CTSLCTSBCTSSCTSK
SCHEMBL4699567 0.78 CTSK (0.44) CTSLCTSBCTSSCTSKKDR
SCHEMBL4703317 0.77 HRH3 (0.35) HRH3CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed