SCHEMBL4704688

SCHEMBL4704688

CC(C)C[C@@H](C(N)=O)N(CC#N)c1cscc1-c1ccc(CN(C)C)cc1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
HRH3 Q9Y5N1 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
CHUK O15111 1/20 0.31
INSR P06213 1/20 0.31
MAPK8 P45983 1/20 0.31
CAMKK2 Q96RR4 1/20 0.31
IKBKE Q14164 1/20 0.31
TBK1 Q9UHD2 1/20 0.31
LGMN Q99538 1/20 0.31
ACVR1 Q04771 1/20 0.31
PARP1 P09874 1/20 0.30
LTB4R2 Q9NPC1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703317 0.91 HRH3 (0.35) CTSLCTSBCTSSCTSKHRH3
SCHEMBL4703269 0.89 ATP4A (0.36) CTSLCTSSCTSKCHUKINSR
SCHEMBL4704896 0.88 CTSK (0.34) CTSLCTSBCTSSCTSK
SCHEMBL4703612 0.87 CTSS (0.34) CTSLCTSBCTSSCTSK
SCHEMBL4701830 0.86 CTSK (0.37) CTSLCTSBCTSSCTSK
SCHEMBL4703639 0.86 CTSK (0.36) CTSLCTSBCTSSCTSK
SCHEMBL4701072 0.85 PDCD1 (0.35) CTSLCTSBCTSSCTSK
SCHEMBL4703746 0.84 OPRM1 (0.37) CTSLCTSBCTSSCTSKHRH3
SCHEMBL4699887 0.83 CTSS (0.34) CTSLCTSBCTSSCTSK
SCHEMBL4699471 0.82 KCNH2 (0.36) CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed