SCHEMBL4700986

SCHEMBL4700986

CCOc1cc(CN(c2ncc(-c3ccc(C(N)=O)cc3)cn2)C2CCNCC2)ccc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.41
SLC6A4 P31645 3/20 0.41
SLC6A3 Q01959 3/20 0.41
FYN P06241 1/20 0.39
AOC3 Q16853 2/20 0.37
CHEK2 O96017 2/20 0.37
CHEK1 O14757 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
KCNH2 Q12809 2/20 0.36
GAA P10253 2/20 0.35
MAP4K4 O95819 1/20 0.34
SSTR5 P35346 2/20 0.34
MAP3K11 Q16584 1/20 0.34
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
TACR1 P25103 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703982 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3AOC3CHEK2
SCHEMBL4702295 0.91 REN (0.42) SLC6A2SLC6A4SLC6A3FYNAOC3
SCHEMBL4704666 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3AOC3KCNH2
SCHEMBL4705165 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3AOC3KCNH2
SCHEMBL3977612 0.87 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3KDM4EALDH1A1
SCHEMBL3973372 0.80 RXRA (0.41) SLC6A2SLC6A4SLC6A3KDM4EALDH1A1
SCHEMBL3971901 0.78 SSTR5 (0.43) SLC6A2SLC6A4SLC6A3KCNH2SSTR5
SCHEMBL3972925 0.78 MAPK1 (0.44) SLC6A2SLC6A4SLC6A3ALDH1A1KCNH2
SCHEMBL3973812 0.77 SSTR5 (0.38) SLC6A2SLC6A4SLC6A3KDM4EKCNH2
SCHEMBL3972873 0.77 SLC6A9 (0.37) SLC6A2SLC6A4SLC6A3KCNH2SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed