SCHEMBL4702295

SCHEMBL4702295

CCOc1cc(CN(c2ncc(-c3ccc(C(N)=O)cc3)cn2)C2CCNCC2)ccc1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 3/20 0.42
MAPK1 P28482 1/20 0.42
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
CHEK1 O14757 1/20 0.39
CHEK2 O96017 1/20 0.39
FYN P06241 2/20 0.38
STK17B O94768 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
AOC3 Q16853 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703982 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3CHEK2MKNK1
SCHEMBL4700986 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3CHEK1CHEK2
SCHEMBL4704666 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3AOC3
SCHEMBL4705165 0.91 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3AOC3
SCHEMBL3972925 0.87 MAPK1 (0.44) RENMAPK1SLC6A2SLC6A4SLC6A3
SCHEMBL3973856 0.81 L3MBTL1 (0.47) RENL3MBTL1ALDH1A1MAPTSMN1; SMN2
SCHEMBL3973369 0.81 REN (0.43) RENMAPK1SLC6A2SLC6A4SLC6A3
SCHEMBL3977361 0.80 REN (0.47) RENMAPK1SLC6A2SLC6A4SLC6A3
SCHEMBL3974286 0.80 REN (0.43) RENL3MBTL1ALDH1A1MAPTSMN1; SMN2
SCHEMBL3973371 0.79 L3MBTL1 (0.53) RENSLC6A2SLC6A4SLC6A3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110340-A2 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed