SCHEMBL4701677

SCHEMBL4701677

Nc1cccc(-n2cnc3c(=O)nc(-c4ccc(Br)cc4)n(-c4ccc(Cl)cc4)c32)c1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.39
XDH P47989 3/20 0.38
MCHR1 Q99705 8/20 0.38
GRM1 Q13255 2/20 0.33
PTGS2 P35354 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5611764 0.88 DHFR (0.43) DHFRXDHMCHR1GRM1PTGS2
SCHEMBL4704498 0.86 MCHR1 (0.38) DHFRXDHMCHR1GRM1PTGS2
SCHEMBL4704274 0.85 KDM4E (0.41) MCHR1MAPTMEN1KMT2A
SCHEMBL4169089 0.85 XDH (0.44) DHFRXDHMCHR1GRM1RXFP1
SCHEMBL4700676 0.84 MCHR1 (0.37) DHFRXDHMCHR1GRM1PTGS2
SCHEMBL5612513 0.80 GRM1 (0.46) XDHMCHR1GRM1PTGS2MAPT
SCHEMBL5611504 0.78 AOC3 (0.44) XDHMCHR1GRM1PTGS2MEN1
SCHEMBL4702957 0.77 PTGS2 (0.39) MCHR1GRM1PTGS2
SCHEMBL5611544 0.76 GRM1 (0.40) XDHMCHR1GRM1PTGS2MEN1
SCHEMBL1689154 0.76 MCHR1 (0.39) XDHMCHR1GRM1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1999132-A1 AZOLOPYRIMIDINES AS INHIBITORS OF CANNABINOID 1 ACTIVITY IRM, LLC (BM) 2008-12-10 EP disclosed
WO-2007120454-A1 AZOLOPYRIMIDINES AS INHIBITORS OF CANNABINOID 1 ACTIVITY IRM LLC (BM) 2007-10-25 WO disclosed