SCHEMBL4708285

SCHEMBL4708285

Cc1cc(C(=O)c2ccccc2Cl)c(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2C2CC2)nn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 9/20 0.38
RORB Q92753 5/20 0.37
RORC P51449 3/20 0.37
TACR1 P25103 1/20 0.36
ROCK2 O75116 2/20 0.36
PIM1 P11309 2/20 0.36
PRKACA P17612 2/20 0.36
CDK2 P24941 2/20 0.36
AURKA O14965 1/20 0.36
CHUK O15111 1/20 0.36
MAPK13 O15264 1/20 0.36
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
CHEK2 O96017 1/20 0.36
PRKCG P05129 1/20 0.36
CDK1 P06493 1/20 0.36
FGFR1 P11362 1/20 0.36
MARK3 P27448 1/20 0.36
MAPK1 P28482 1/20 0.36
AKT1 P31749 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707181 0.88 RORB (0.40) CDC7RORBRORCTACR1ROCK2
SCHEMBL4705642 0.86 RORB (0.40) CDC7RORBRORCTACR1ROCK2
SCHEMBL4705944 0.85 TACR1 (0.39) RORBRORCTACR1GAAKCNJ6
SCHEMBL4708690 0.85 RORB (0.40) CDC7RORBRORCTACR1GAA
SCHEMBL4706783 0.83 RORB (0.38) CDC7RORBRORCTACR1MAPK1
SCHEMBL4708438 0.82 CDC7 (0.41) CDC7TACR1ROCK2PIM1PRKACA
SCHEMBL4707207 0.82 RORB (0.40) RORBRORCTACR1GAA
SCHEMBL4707706 0.81 IDH1 (0.42) RORBRORCTACR1KDRCRHR1
SCHEMBL4707926 0.80 P2RX7 (0.36) RORBRORCTACR1GAA
SCHEMBL4706857 0.80 CDC7 (0.37) CDC7RORBRORCTACR1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed