SCHEMBL4710002

SCHEMBL4710002

COc1cc(C(=O)[C@H]2C(=O)c3cc(C(=O)NNC(=O)OC(C)(C)C)ccc3OC23CCNCC3)nc2c(OC)cccc12

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.36
ACACA Q13085 1/20 0.36
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708596 0.86 ACACA (0.36) ACACBACACALMNATP53
SCHEMBL4710103 0.84 ACACA (0.37) ACACBACACA
SCHEMBL4708583 0.82 XIAP (0.39) ACACBACACALMNA
SCHEMBL4707267 0.82 ACACA (0.38) ACACBACACA
SCHEMBL4707168 0.82 MEN1 (0.36) ACACBACACALMNA
SCHEMBL4708996 0.81 ACACA (0.35) ACACBACACA
SCHEMBL4759738 0.80 HTR7 (0.38) ACACBACACA
SCHEMBL4760214 0.80 ACACA (0.34) ACACBACACA
SCHEMBL4709980 0.79 ACACA (0.36) ACACBACACA
SCHEMBL4759789 0.78 TNKS (0.34) ACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910375-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS Merck & Co., Inc. (US) 2008-04-16 EP disclosed
WO-2007011809-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK & CO., INC. (US) 2007-01-25 WO disclosed