SCHEMBL4708975

SCHEMBL4708975

CC(C)(C)OC(=O)ON1CCN(CCCSc2cccs2)CC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
DRD2 P14416 5/20 0.35
SIGMAR1 Q99720 3/20 0.35
ACKR3 P25106 2/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HRH2 P25021 1/20 0.34
HRH1 P35367 1/20 0.34
KCNH2 Q12809 3/20 0.34
HTR1A P08908 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3766890 0.85 ACKR3 (0.48) SIGMAR1ACKR3HRH2HRH1
SCHEMBL8618331 0.71 GPR119 (0.49) KDM4E
SCHEMBL249745 0.70 DRD2 (0.36) DRD2SIGMAR1
SCHEMBL3781095 0.70 CYP1A2 (0.49) KDM4EALDH1A1DRD2SIGMAR1HRH2
SCHEMBL8316805 0.67 CCNB2 (0.48) KDM4EALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL9141640 0.66 SIGMAR1 (0.55) ALDH1A1DRD2SIGMAR1HTR1A
SCHEMBL1444698 0.65 MPO (0.56) KDM4EALDH1A1MEN1KMT2A
SCHEMBL5228089 0.65 SMN1; SMN2 (0.53) KDM4EALDH1A1SIGMAR1ACKR3MEN1
SCHEMBL7612299 0.65 TACR1 (0.35) DRD2SIGMAR1
SCHEMBL688938 0.64 HSD17B10 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943222-A1 ANTIBACTERIAL ACTIVE 5-CHINOLIN DERIVATIVE Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2008-07-16 EP disclosed
WO-2007042325-A1 ANTIBACTERIAL ACTIVE 5-CHINOLIN DERIVATIVE Morphochem Aktiengesellschaft für kombinatorische Chemie (DE) 2007-04-19 WO disclosed