SCHEMBL4710667

SCHEMBL4710667

CCN(c1c(F)cccc1F)C1CN(C(=O)O)C1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.38
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
OXTR P30559 1/20 0.35
NOTUM Q6P988 1/20 0.34
HCRTR1 O43613 4/20 0.34
HCRTR2 O43614 4/20 0.34
HPGD P15428 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4713873 0.78 HRH3 (0.38) OPRM1ALDH1A1
SCHEMBL4715539 0.75 ALDH1A1 (0.41) ALDH1A1NOTUMHPGDLMNA
SCHEMBL4716542 0.74 LMNA (0.41) OPRM1ALDH1A1LMNA
SCHEMBL4713689 0.74 SMN1; SMN2 (0.38) OPRM1ALDH1A1HPGD
SCHEMBL4714369 0.73 OPRM1 (0.42) OPRM1KDM4EALDH1A1NOTUMHPGD
SCHEMBL4714471 0.73 OXTR (0.38) ALDH1A1OXTR
SCHEMBL4713625 0.72 CYP2D6 (0.38) KDM4EALDH1A1OXTRHPGD
SCHEMBL4714260 0.71 MEN1 (0.43) KDM4EALDH1A1LMNA
SCHEMBL4716576 0.70 ALDH1A1 (0.40) OPRM1KDM4EALDH1A1HPGDLMNA
SCHEMBL1575172 0.70 KDM4E (0.58) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933830-A1 ANTAGONISTS OF SNS SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-06-25 EP disclosed
WO-2007007057-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed