SCHEMBL4715545

SCHEMBL4715545

CC(NC(=O)C(=O)c1c[nH]c2ccccc12)c1ccccc1N1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
KMT2A Q03164 1/20 0.54
KDM4E B2RXH2 1/20 0.54
LMNA P02545 1/20 0.54
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
PKM P14618 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4715552 0.76 RAB9A (0.58) ALDH1A1KMT2AKDM4ELMNANPC1
SCHEMBL20746151 0.75 ALDH1A1 (0.51) ALDH1A1KMT2ALMNAPKM
SCHEMBL30712073 0.74 ALOX5 (0.63) KMT2ANPC1RAB9A
SCHEMBL19459867 0.74 ALOX5 (0.63) KMT2ANPC1RAB9A
SCHEMBL4715549 0.73 ALDH1A1 (0.55) ALDH1A1KMT2AKDM4ELMNANPC1
SCHEMBL1558423 0.71 ALDH1A1 (1.00) ALDH1A1KMT2AKDM4ELMNARAB9A
SCHEMBL393338 0.69 CFTR (0.57) ALDH1A1KMT2APKM
SCHEMBL1413396 0.68 ALDH1A1 (0.55) ALDH1A1KMT2AKDM4ELMNA
SCHEMBL11921542 0.68 CFTR (0.68) ALDH1A1KMT2ANPC1RAB9A
SCHEMBL20181880 0.68 ALDH1A1 (0.75) ALDH1A1KMT2AKDM4ELMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933831-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals, Inc. (US) 2008-06-25 EP claimed
WO-2007044560-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-04-19 WO claimed