SCHEMBL4715552

SCHEMBL4715552

O=C(NCCc1ccccc1N1CCOCC1)C(=O)c1c[nH]c2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.58
NPC1 O15118 1/20 0.58
ALDH1A1 P00352 4/20 0.54
KMT2A Q03164 4/20 0.54
IGF1R P08069 1/20 0.54
LMNA P02545 2/20 0.54
KDM4E B2RXH2 1/20 0.54
POLB P06746 3/20 0.53
MEN1 O00255 3/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HPGD P15428 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
GABRP O00591 3/20 0.51
GABRD O14764 3/20 0.51
GABRA1 P14867 3/20 0.51
GABRB1 P18505 3/20 0.51
GABRG2 P18507 3/20 0.51
GABRB3 P28472 3/20 0.51
GABRA5 P31644 3/20 0.51
GABRA3 P34903 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26090898 0.79 RAB9A (0.76) RAB9ANPC1ALDH1A1KMT2AIGF1R
SCHEMBL4715545 0.76 ALDH1A1 (0.54) RAB9ANPC1ALDH1A1KMT2ALMNA
SCHEMBL4760802 0.74 RAB9A (1.00) RAB9ANPC1ALDH1A1KMT2AIGF1R
SCHEMBL30712063 0.72 NPC1 (0.71) RAB9ANPC1KMT2AIGF1RPOLB
SCHEMBL1558423 0.71 ALDH1A1 (1.00) RAB9AALDH1A1KMT2ALMNAKDM4E
SCHEMBL20267059 0.70 HPGD (0.61) ALDH1A1KMT2ALMNAKDM4EMEN1
SCHEMBL31060147 0.70 POLB (0.73) RAB9ANPC1KMT2AIGF1RPOLB
SCHEMBL3722135 0.70 ALDH1A1 (0.61) ALDH1A1KMT2ALMNAKDM4EMEN1
SCHEMBL30712070 0.69 GABRP (0.72) RAB9ANPC1KMT2AIGF1RPOLB
SCHEMBL393338 0.69 CFTR (0.57) ALDH1A1KMT2APOLBMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933831-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals, Inc. (US) 2008-06-25 EP claimed
WO-2007044560-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-04-19 WO claimed