SCHEMBL4718491

SCHEMBL4718491

COc1ccc(-c2ccc3c(c2)N=C(N)N(Cc2c(OC)cccc2OC)C3)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 9/20 0.40
ABCB1 P08183 6/20 0.38
ABCC1 P33527 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
ADORA1 P30542 1/20 0.36
DRD4 P21917 2/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
SLC6A2 P23975 1/20 0.35
HTR2C P28335 1/20 0.35
SLC6A4 P31645 1/20 0.35
OPRK1 P41145 1/20 0.35
HTR2B P41595 1/20 0.35
HTR5A P47898 1/20 0.35
SLC6A3 Q01959 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL3206340 0.94 CTSD (0.39) CTSDABCB1ABCC1BACE1
SCHEMBL4715532 0.92 CTSD (0.48) CTSDABCB1DRD4HTR1AADRA2A
SCHEMBL4716520 0.90 GRIN2B (0.42) CTSDBACE1
Acetic Acid SCHEMBL3263693 0.88 CTSD (0.44) CTSDDRD4HTR1AADRA2AADRA2B
SCHEMBL4716955 0.85 HCRTR1 (0.42) CTSDBACE1
SCHEMBL4719286 0.84 CTSD (0.43) CTSD
SCHEMBL4714576 0.83 APLNR (0.38) CTSDADORA1DRD4DRD2DRD3
SCHEMBL3209339 0.83 CTSD (0.57) CTSDDRD4ADRA2ADRD2
SCHEMBL3198015 0.83 CTSD (0.42) CTSD
SCHEMBL4714175 0.81 SIGMAR1 (0.44) CTSDADRA2BHTR5ASIGMAR1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917245-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS Abbott GmbH & Co. KG (DE) 2008-05-07 EP disclosed
WO-2007022946-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS ABBOTT GMBH & CO. KG (DE) 2007-03-01 WO disclosed