SCHEMBL4715532

SCHEMBL4715532

COc1cccc(OC)c1CN1Cc2ccc(-c3ccccc3)cc2N=C1N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 4/20 0.48
DRD4 P21917 4/20 0.38
TMEM97 Q5BJF2 3/20 0.38
SIGMAR1 Q99720 3/20 0.38
HTR2C P28335 3/20 0.38
HTR1A P08908 2/20 0.38
HTR2B P41595 2/20 0.38
SLC6A3 Q01959 2/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
OPRK1 P41145 1/20 0.38
HTR5A P47898 1/20 0.38
HCRTR1 O43613 3/20 0.36
HCRTR2 O43614 3/20 0.36
DRD3 P35462 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM3 P20309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL3263693 0.95 CTSD (0.44) CTSDDRD4TMEM97SIGMAR1HTR2C
SCHEMBL4718491 0.92 CTSD (0.40) CTSDDRD4TMEM97SIGMAR1HTR2C
Acetic Acid SCHEMBL3206340 0.89 CTSD (0.39) CTSDABCB1BACE1KDM4EALDH1A1
SCHEMBL4716955 0.89 HCRTR1 (0.42) CTSDHCRTR1HCRTR2BACE1
SCHEMBL4716520 0.87 GRIN2B (0.42) CTSDHCRTR1HCRTR2BACE1
Acetic Acid SCHEMBL3212866 0.86 MKNK1 (0.44) CTSDHCRTR1HCRTR2BACE1
SCHEMBL4719286 0.85 CTSD (0.43) CTSDKDM4EALDH1A1
SCHEMBL4714175 0.85 SIGMAR1 (0.44) CTSDSIGMAR1ADRA2BHTR5ABACE1
SCHEMBL4714576 0.84 APLNR (0.38) CTSDDRD4DRD3DRD2KDM4E
SCHEMBL3198015 0.84 CTSD (0.42) CTSDKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917245-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS Abbott GmbH & Co. KG (DE) 2008-05-07 EP disclosed
WO-2007022946-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS ABBOTT GMBH & CO. KG (DE) 2007-03-01 WO disclosed