SCHEMBL4719286

SCHEMBL4719286

COc1cccc(OC)c1CN1Cc2ccc(C)cc2N=C1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 9/20 0.43
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 1/20 0.34
UGCG Q16739 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
SPIN1 Q9Y657 1/20 0.32
TACR1 P25103 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
MDM2 Q00987 1/20 0.32
MEN1 O00255 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL3207125 0.94 CTSD (0.39) CTSDSMN1; SMN2NPC1TP53GAA
SCHEMBL3209339 0.87 CTSD (0.57) CTSDALDH1A1CYP3A4KDM4E
SCHEMBL3198015 0.87 CTSD (0.42) CTSDALDH1A1SPIN1KDM4E
SCHEMBL4715532 0.85 CTSD (0.48) CTSDALDH1A1KDM4E
SCHEMBL4714175 0.85 SIGMAR1 (0.44) CTSDALDH1A1TACR1KDM4EMAPK1
SCHEMBL4718491 0.84 CTSD (0.40) CTSD
SCHEMBL4718254 0.82 CTSD (0.39) CTSDGAAALDH1A1KDM4ELMNA
Acetic Acid SCHEMBL3263693 0.81 CTSD (0.44) CTSDGAAALDH1A1KDM4ELMNA
SCHEMBL4714576 0.81 APLNR (0.38) CTSDSMN1; SMN2NPC1TP53TSHR
SCHEMBL4716955 0.81 HCRTR1 (0.42) CTSDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917245-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS Abbott GmbH & Co. KG (DE) 2008-05-07 EP disclosed
WO-2007022946-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS ABBOTT GMBH & CO. KG (DE) 2007-03-01 WO disclosed