SCHEMBL4720655

SCHEMBL4720655

COC(=O)c1cc(-c2cc(C)cc(CO)c2)nn(-c2cc(Br)ccc2C(F)(F)F)c1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 3/20 0.34
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
LMNA P02545 1/20 0.33
NOTUM Q6P988 1/20 0.33
CYP46A1 Q9Y6A2 1/20 0.32
MET P08581 1/20 0.32
PTGER1 P34995 1/20 0.32
MBOAT4 Q96T53 1/20 0.32
SLC6A3 Q01959 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PTGER4 P35408 1/20 0.31
RET P07949 1/20 0.31
PRKX P51817 1/20 0.31
TAOK1 Q7L7X3 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723668 0.75 TACR1 (0.36) NTRK1LMNA
SCHEMBL4719000 0.68 PTK2 (0.36) NTRK1MEN1KMT2A
SCHEMBL4720918 0.66 GPR119 (0.33)
SCHEMBL4722667 0.66 AR (0.34) NTRK1LMNAPTGER1SMN1; SMN2RET
SCHEMBL4720784 0.66 PDE4A (0.38)
SCHEMBL155135 0.65 NOTUM (0.58) LMNANOTUMMBOAT4SLC6A3SMN1; SMN2
SCHEMBL30736877 0.65 NOTUM (0.58) LMNANOTUMMBOAT4SLC6A3SMN1; SMN2
SCHEMBL19940155 0.64 SLC6A3 (0.55) LMNACYP46A1SLC6A3KDM4EKMT2A
SCHEMBL4721524 0.62 BRD4 (0.33)
SCHEMBL516822 0.62 NOTUM (0.54) NOTUMSLC6A3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed