SCHEMBL4722103

SCHEMBL4722103

COc1cc(OC)cc(-c2nn(-c3ccccc3C(F)(F)F)c(=O)c3c2CCN3)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.35
SLC16A3 O15427 1/20 0.35
SLC16A1 P53985 1/20 0.35
MGLL Q99685 1/20 0.35
PHGDH O43175 1/20 0.34
CNR1 P21554 2/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
MAPT P10636 3/20 0.33
GRM7 Q14831 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
CNR2 P34972 1/20 0.33
CRHR1 P34998 2/20 0.33
TP53 P04637 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
TEK Q02763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720876 0.89 CYP11B1 (0.33) MAPTGRM7ALDH1A1ALPLALPI
SCHEMBL14101738 0.88 LRRK2 (0.33) GRM7ALPLALPI
SCHEMBL4719266 0.88 LRRK2 (0.33) GRM7CRHR1ALPLALPI
SCHEMBL4764976 0.88 CNR1 (0.34) CNR1GRM7CNR2ALPLALPI
SCHEMBL4724987 0.85 F10 (0.40) MAPTPOLBALDH1A1
SCHEMBL4724951 0.84 NTRK1 (0.32) MAPTGRM7MEN1GAAKMT2A
SCHEMBL4720114 0.84 PDE4A (0.47) L3MBTL1SLC16A3SLC16A1MGLLPHGDH
SCHEMBL4721216 0.83 F10 (0.32) MAPTALPLALPI
SCHEMBL4718926 0.81 F10 (0.32) GRM7
SCHEMBL4724753 0.81 BRAF (0.33) GAAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed