SCHEMBL4721152

SCHEMBL4721152

CNC(=O)NN(Cc1ccc(-c2ccccc2)cc1)C(=O)c1ccc(OC(C)C)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 1/20 0.52
S1PR1 P21453 4/20 0.44
S1PR3 Q99500 2/20 0.44
KIFC1 Q9BW19 1/20 0.42
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
P2RX3 P56373 1/20 0.39
CSNK2A1 P68400 2/20 0.38
RORC P51449 1/20 0.38
KMO O15229 2/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
MAP4K4 O95819 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
S1PR5 Q9H228 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4521076 0.91 CENPE (0.47) CENPES1PR1S1PR3KIFC1MEN1
SCHEMBL4719991 0.89 CENPE (0.48) CENPES1PR1S1PR3KIFC1MEN1
SCHEMBL4722528 0.89 CENPE (0.53) CENPEMEN1KMT2AP2RX3RORC
SCHEMBL4720776 0.88 CENPE (0.44) CENPES1PR1S1PR3KIFC1MEN1
SCHEMBL4718072 0.88 CENPE (0.46) CENPEMEN1KMT2AP2RX3CYP1A2
SCHEMBL2103268 0.85 CENPE (0.56) CENPES1PR1S1PR3KIFC1MEN1
SCHEMBL4717871 0.84 CENPE (0.43) CENPE
SCHEMBL4720908 0.84 MEN1 (0.47) CENPEMEN1KMT2ACYP1A2CYP2C9
SCHEMBL4720150 0.84 PTGES (0.46) CENPEKMT2AP2RX3MAPTSMN1; SMN2
SCHEMBL2104964 0.82 CENPE (0.53) CENPES1PR1S1PR3KIFC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP disclosed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed