SCHEMBL4720908

SCHEMBL4720908

CNC(=O)NN(Cc1ccc(OCc2ccccc2)c(OC)c1)C(=O)c1ccc(OC(C)C)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
TRPM8 Q7Z2W7 1/20 0.45
RAF1 P04049 4/20 0.44
MAP2K1 Q02750 4/20 0.44
CENPE Q02224 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
APP P05067 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718072 0.89 CENPE (0.46) MEN1KMT2ACENPEKDM4ECYP1A2
SCHEMBL4720150 0.88 PTGES (0.46) KMT2ACENPENPC1RAB9AHPGD
SCHEMBL2104713 0.87 CENPE (0.48) MEN1KMT2ATRPM8RAF1MAP2K1
SCHEMBL4721152 0.84 CENPE (0.52) MEN1KMT2ACENPESMN1; SMN2CYP1A2
SCHEMBL4722528 0.81 CENPE (0.53) MEN1KMT2ACENPENPC1RAB9A
SCHEMBL4720776 0.80 CENPE (0.44) MEN1KMT2ACENPEHPGDKDM4E
SCHEMBL4720907 0.80 TRPM8 (0.50) MEN1KMT2ATRPM8RAF1MAP2K1
SCHEMBL13584065 0.79 MEN1 (0.51) MEN1KMT2ATRPM8RAF1MAP2K1
SCHEMBL4721237 0.79 SPHK2 (0.44) KMT2ACENPEKDM4ECYP1A2CYP2C9
SCHEMBL13711251 0.77 MEN1 (0.47) MEN1KMT2ATRPM8RAF1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP claimed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO claimed
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP disclosed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed