SCHEMBL4722534

SCHEMBL4722534

COc1cc(OC)cc(-c2cn(-c3cc(N4CC(CO)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3CC(N)=O)c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 1/20 0.34
F10 P00742 2/20 0.32
WDR5 P61964 6/20 0.31
CXCR3 P49682 2/20 0.31
CMA1 P23946 1/20 0.30
AKR1B10 O60218 1/20 0.30
AKR1C4 P17516 1/20 0.30
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30
AKR1C1 Q04828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719537 0.94 S1PR1 (0.35) F10CXCR3CMA1AKR1C4AKR1C3
SCHEMBL4719467 0.91 WDR5 (0.34) ACVR1WDR5
SCHEMBL4719251 0.90 ACVR1 (0.35) ACVR1F10CXCR3AKR1B10AKR1C4
SCHEMBL4719937 0.87 ACVR1 (0.32) ACVR1WDR5CXCR3AKR1B10AKR1C4
SCHEMBL14101950 0.84 UCHL1 (0.37) ACVR1F10CXCR3CMA1AKR1C4
SCHEMBL4722741 0.81 UCHL1 (0.38) CXCR3CMA1AKR1C4AKR1C3AKR1C2
SCHEMBL4719462 0.81 CXCR3 (0.35) F10CXCR3
SCHEMBL4721143 0.79 SUV39H2 (0.36) WDR5
SCHEMBL4721137 0.79 SUV39H2 (0.36) WDR5
SCHEMBL4721921 0.79 CXCR3 (0.33) F10WDR5CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed