SCHEMBL14101950

SCHEMBL14101950

COc1cccc(-c2cn(-c3cc(N4CC(CO)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3C(N)=O)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.37
USP30 Q70CQ3 1/20 0.37
S1PR1 P21453 1/20 0.36
CXCR3 P49682 1/20 0.34
HDAC6 Q9UBN7 2/20 0.33
CYP2C9 P11712 1/20 0.33
AKR1C4 P17516 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
DGAT2 Q96PD7 3/20 0.33
F10 P00742 1/20 0.33
RBP4 P02753 1/20 0.33
BRD4 O60885 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32
ABL2 P42684 1/20 0.32
MCHR1 Q99705 1/20 0.32
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722741 0.94 UCHL1 (0.38) UCHL1USP30S1PR1CXCR3HDAC6
SCHEMBL4719251 0.94 ACVR1 (0.35) CXCR3AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL4719537 0.90 S1PR1 (0.35) UCHL1USP30S1PR1CXCR3HDAC6
SCHEMBL4719937 0.86 ACVR1 (0.32) CXCR3AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL4723936 0.85 SMN1; SMN2 (0.35) UCHL1USP30S1PR1CXCR3HDAC6
SCHEMBL4722534 0.84 ACVR1 (0.34) CXCR3AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL4719467 0.81 WDR5 (0.34) KMT2AACVR1
SCHEMBL4722281 0.81 LIPG (0.38) F10RBP4
SCHEMBL4722284 0.81 LIPG (0.38) F10RBP4
SCHEMBL4721394 0.80 F10 (0.33) CXCR3F10RBP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed