SCHEMBL4722741

SCHEMBL4722741

COc1cccc(-c2cn(-c3cc(N4CC(CO)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3C(=O)O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.38
USP30 Q70CQ3 1/20 0.38
S1PR1 P21453 1/20 0.38
AKR1C4 P17516 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35
CXCR3 P49682 1/20 0.34
HDAC6 Q9UBN7 2/20 0.34
CYP2C9 P11712 1/20 0.34
DGAT2 Q96PD7 5/20 0.34
FFAR1 O14842 3/20 0.33
CMA1 P23946 1/20 0.33
MCHR1 Q99705 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
GRM5 P41594 1/20 0.32
AKT1 P31749 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14101950 0.94 UCHL1 (0.37) UCHL1USP30S1PR1AKR1C4AKR1C3
SCHEMBL4719537 0.88 S1PR1 (0.35) UCHL1USP30S1PR1AKR1C4AKR1C3
SCHEMBL4719251 0.87 ACVR1 (0.35) AKR1C4AKR1C3AKR1C2AKR1C1CXCR3
SCHEMBL4719937 0.87 ACVR1 (0.32) AKR1C4AKR1C3AKR1C2AKR1C1CXCR3
SCHEMBL4719467 0.82 WDR5 (0.34) KMT2A
SCHEMBL4722534 0.81 ACVR1 (0.34) AKR1C4AKR1C3AKR1C2AKR1C1CXCR3
SCHEMBL4723936 0.79 SMN1; SMN2 (0.35) UCHL1USP30S1PR1CXCR3HDAC6
SCHEMBL4722418 0.77 PDCD1 (0.32) UCHL1USP30LMNAAKT1
SCHEMBL4720389 0.77 MTNR1A (0.40) UCHL1USP30S1PR1CXCR3DGAT2
SCHEMBL4720392 0.77 MTNR1A (0.40) UCHL1USP30S1PR1CXCR3DGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed