SCHEMBL4725920

SCHEMBL4725920

Cc1ncc(NC(=O)c2cc(C#N)cc(C(C)(C)C)c2)cc1-c1ccc(C(=O)NCC2CCCO2)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 3/20 0.48
CYP2C9 P11712 1/20 0.48
MAPK14 Q16539 1/20 0.48
NAMPT P43490 3/20 0.46
TAAR1 Q96RJ0 1/20 0.45
LMNA P02545 2/20 0.44
ALDH1A1 P00352 1/20 0.44
ALOX12 P18054 1/20 0.44
ATM Q13315 1/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
HPGD P15428 5/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HTT P42858 1/20 0.44
POLB P06746 2/20 0.44
CYP1A2 P05177 1/20 0.44
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4728308 0.91 EGLN1 (0.48) EGLN1NAMPTTAAR1LMNAALDH1A1
SCHEMBL4728367 0.89 MAPK14 (0.50) CYP2C9MAPK14TAAR1LMNAALDH1A1
SCHEMBL4727468 0.88 MAPK14 (0.47) EGLN1MAPK14NAMPT
SCHEMBL4728099 0.85 RAF1 (0.41) EGLN1MAPK14
SCHEMBL4725917 0.84 RAF1 (0.44)
SCHEMBL4726798 0.83 RAF1 (0.42)
SCHEMBL4729070 0.83 IKBKB (0.43) EGLN1MAPK14ALDH1A1KMT2AMEN1
SCHEMBL4729206 0.82 RAF1 (0.47) EGLN1MAPK14
SCHEMBL4727147 0.82 MAPK14 (0.48) EGLN1MAPK14KMT2AMEN1
SCHEMBL4729551 0.82 RAF1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed