SCHEMBL4735258

SCHEMBL4735258

CCN(CC)c1cccc(CN(C(=O)c2ccco2)c2ccc(Cl)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
LMNA P02545 5/20 0.46
TSHR P16473 4/20 0.46
MAPT P10636 3/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 5/20 0.46
MEN1 O00255 4/20 0.46
RAD52 P43351 2/20 0.44
CNR2 P34972 1/20 0.43
POLB P06746 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALOX15 P16050 1/20 0.41
TP53 P04637 2/20 0.41
NPC1 O15118 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4734930 0.81 ALDH1A1 (0.45) ALDH1A1LMNAMAPTKMT2AMEN1
SCHEMBL8190064 0.80 CYP3A4 (0.42) LMNATSHRMAPTKMT2AMEN1
SCHEMBL3818747 0.79 CNR2 (0.47) ALDH1A1LMNAMAPTHTTCNR2
SCHEMBL8184199 0.78 MAPK14 (0.44) MAPTCNR2CYP3A4TP53
SCHEMBL4739106 0.78 NPC1 (0.41) MAPTKMT2AMEN1CNR2POLB
SCHEMBL4738668 0.78 CNR2 (0.40) MAPTCNR2CYP3A4
SCHEMBL4733577 0.78 TLR7 (0.40) ALDH1A1LMNAMAPTCNR2CYP3A4
SCHEMBL3824123 0.78 CNR1 (0.41) ALDH1A1LMNAMAPTCNR2POLB
SCHEMBL4733672 0.77 ALDH1A1 (0.44) ALDH1A1LMNACNR2SMN1; SMN2
SCHEMBL4736765 0.77 CYP19A1 (0.43) MAPTHTTCNR2CYP1A2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed