SCHEMBL4736402

SCHEMBL4736402

CC(C)c1cc2c(cc1S(=O)(=O)NC1Cc3ccccc3C1)S(=O)(=O)c1cc(F)ccc1CC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.38
HTR7 P34969 6/20 0.38
DRD2 P14416 3/20 0.38
HTR6 P50406 3/20 0.38
PSEN1 P49768 4/20 0.37
PSEN2 P49810 4/20 0.37
APH1B Q8WW43 4/20 0.37
NCSTN Q92542 4/20 0.37
APH1A Q96BI3 4/20 0.37
PSENEN Q9NZ42 4/20 0.37
GRIA2 P42262 4/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NR1H2 P55055 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
ADRA1D P25100 1/20 0.35
HTR2A P28223 1/20 0.35
ADRA1A P35348 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4735405 0.88 HTR1A (0.39) HTR1AHTR7DRD2HTR6MEN1
SCHEMBL4731657 0.85 HTR1A (0.38) HTR1AHTR7DRD2HTR6PSEN1
SCHEMBL4730503 0.80 SMN1; SMN2 (0.47) KMT2A
SCHEMBL4732619 0.79 TAAR1 (0.43) KMT2A
SCHEMBL4734310 0.77 AKR1C3 (0.38) HTR1AHTR7DRD2HTR6HTR2A
SCHEMBL4733242 0.77 TDP1 (0.42) KMT2A
SCHEMBL4732992 0.77 CA1 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4731425 0.77 KMT2A (0.40) HTR1AHTR7DRD2HTR6MEN1
SCHEMBL4733452 0.76 CNR2 (0.39) HTR1AHTR7DRD2HTR6MEN1
SCHEMBL4731644 0.75 ACHE (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO claimed
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed