SCHEMBL4737014

SCHEMBL4737014

O=C(c1ccnnc1)N(Cc1ccc(N2CCNCC2)nc1)c1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 6/20 0.42
HDAC3 O15379 5/20 0.42
MAPK14 Q16539 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MAPKAPK2 P49137 3/20 0.39
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
ME2 P23368 1/20 0.38
ME1 P48163 1/20 0.38
ME3 Q16798 1/20 0.38
MLNR O43193 2/20 0.38
CXCR2 P25025 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
HPGDS O60760 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4735426 0.90 OPRM1 (0.43) MAPK14OPRM1OPRK1ME2ME1
SCHEMBL4738924 0.89 OPRM1 (0.40) MAPK14HDAC10OPRM1OPRK1ME2
SCHEMBL4735517 0.88 MAPK14 (0.38) MAPK14OPRM1OPRK1ME2ME1
SCHEMBL4733795 0.88 KDM4E (0.51) MAPK14OPRM1OPRK1ME2ME1
SCHEMBL4737305 0.88 DRD4 (0.45) MAPK14CXCR2KDM4EALDH1A1TSHR
SCHEMBL4738909 0.87 TSHR (0.44) MAPK14OPRM1OPRK1ME2ME1
SCHEMBL3826843 0.86 MAPKAPK2 (0.47) HDAC2HDAC3HDAC1HDAC10HDAC6
SCHEMBL4733666 0.85 OPRM1 (0.49) MAPK14OPRM1OPRK1KDM4EALDH1A1
SCHEMBL4738700 0.84 MAPK14 (0.39) MAPK14MLNRCXCR2KDM4EALDH1A1
SCHEMBL4735512 0.84 HRH3 (0.43) MAPK14OPRM1OPRK1ME2ME1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed