SCHEMBL4738700

SCHEMBL4738700

CC1CC(C)CN(c2ccc(CN(C(=O)c3ccnnc3)c3ccc(F)cc3)cn2)C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.39
MLNR O43193 8/20 0.38
CXCR2 P25025 1/20 0.37
CNR2 P34972 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4738924 0.86 OPRM1 (0.40) MAPK14CXCR2KDM4EALDH1A1TSHR
SCHEMBL4735426 0.86 OPRM1 (0.43) MAPK14CXCR2KDM4EALDH1A1TSHR
SCHEMBL4733765 0.85 CNR2 (0.36) MAPK14MLNRCXCR2CNR2KDM4E
SCHEMBL4737014 0.84 HDAC2 (0.42) MAPK14MLNRCXCR2KDM4EALDH1A1
SCHEMBL4735517 0.84 MAPK14 (0.38) MAPK14MLNRCXCR2KDM4EALDH1A1
SCHEMBL4737305 0.83 DRD4 (0.45) MAPK14CXCR2KDM4EALDH1A1TSHR
SCHEMBL4733795 0.83 KDM4E (0.51) MAPK14CXCR2KDM4EALDH1A1TSHR
SCHEMBL4738909 0.83 TSHR (0.44) MAPK14CXCR2KDM4EALDH1A1TSHR
SCHEMBL4735512 0.81 HRH3 (0.43) MAPK14TSHRHSD17B10
SCHEMBL4733666 0.80 OPRM1 (0.49) MAPK14KDM4EALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed