SCHEMBL4737056

SCHEMBL4737056

O=C(O)N(Cc1cccc(NC2CC2)c1)c1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.47
CHRM1 P11229 2/20 0.47
CHRM3 P20309 2/20 0.47
MAPK14 Q16539 1/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
PDK1 Q15118 2/20 0.41
ACHE P22303 1/20 0.40
PTPRB P23467 1/20 0.40
ACKR3 P25106 1/20 0.39
MEP1B Q16820 1/20 0.39
PTGES O14684 1/20 0.39
AGER Q15109 2/20 0.39
MTNR1A P48039 1/20 0.39
UBE2M P61081 1/20 0.39
DCUN1D1 Q96GG9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4738206 0.86 CHRM2 (0.46) CHRM2CHRM1CHRM3MAPK14KDM4E
SCHEMBL3058213 0.84 CHRM1 (0.44) CHRM2CHRM1CHRM3KDM4EACHE
SCHEMBL13090649 0.78 KDM4E (0.45) CHRM2CHRM1CHRM3KDM4EALDH1A1
SCHEMBL3830101 0.76 ALDH1A1 (0.44) CHRM2CHRM1CHRM3MAPK14KDM4E
SCHEMBL19868563 0.73 LOXL2 (0.51) MAPTKDM4EALDH1A1MEP1B
SCHEMBL3824005 0.71 L3MBTL1 (0.47) MAPTKDM4EALDH1A1
SCHEMBL3058780 0.71 CHRM1 (0.44) CHRM2CHRM1CHRM3MAPTALDH1A1
SCHEMBL4237307 0.71 ALDH1A1 (0.54) MAPK14KDM4EALDH1A1TSHR
SCHEMBL28986105 0.70 NPC1 (0.61) ALDH1A1TSHRPDK1
SCHEMBL6831433 0.69 LTB4R2 (0.54) MAPK14PTPRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed