SCHEMBL4737951

SCHEMBL4737951

COc1cc(OC)cc(C(=S)Nc2c(C)cccc2C)c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
GAA P10253 2/20 0.44
NPC1 O15118 4/20 0.44
RAB9A P51151 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HPGD P15428 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPK1 P28482 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HTT P42858 2/20 0.41
ALOX12 P18054 1/20 0.41
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741248 0.81 KDM4E (0.47) ALDH1A1GAARAB9ASMN1; SMN2MAPT
SCHEMBL1817099 0.72 KMT2A (0.53) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL1814123 0.71 LMNA (0.63) GAAMEN1KMT2AL3MBTL1ALOX12
SCHEMBL6935548 0.69 ALDH1A1 (0.65) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL31465658 0.69 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MAPTCYP3A4HPGD
SCHEMBL4739005 0.69 ALDH1A1 (0.65) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL15484311 0.68 LMNA (0.69) ALDH1A1GAANPC1RAB9ASMN1; SMN2
SCHEMBL28466686 0.68 NPC1 (0.69) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL11919007 0.67 FFAR4 (0.41) ALDH1A1MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL31465694 0.67 CES2 (0.55) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008077170-A2 BENZOTHIOAMIDES, AND USE THEREOF FOR RELAXING SMOOTH MUSCLES Universität Wien (AT) 2008-07-03 WO disclosed