SCHEMBL474062

SCHEMBL474062

Cn1c(=O)oc2ccc(CC(c3ccc(Br)cc3C(F)(F)F)C(O)C(F)(F)F)cc21

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.35
KCNJ1 P48048 12/20 0.34
ASAH1 Q13510 2/20 0.34
SIGMAR1 Q99720 1/20 0.32
KMO O15229 1/20 0.32
CMA1 P23946 1/20 0.31
CTSC P53634 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473987 0.89 CYP11B2 (0.35) CYP11B2KCNJ1ASAH1SIGMAR1CTSC
SCHEMBL473924 0.81 CYP11B2 (0.41) CYP11B2
SCHEMBL473947 0.80 MIF (0.36) CYP11B2KCNJ1CTSC
SCHEMBL474137 0.80 MIF (0.36) CYP11B2KCNJ1CTSC
SCHEMBL473926 0.78 KMO (0.39) CYP11B2ASAH1KMO
SCHEMBL474034 0.76 KMO (0.39) CYP11B2KMO
SCHEMBL473936 0.75 CYP11B2 (0.45) CYP11B2KCNJ1CTSC
SCHEMBL474022 0.75 ALDH1A1 (0.38) CYP11B2KCNJ1KMOCMA1
SCHEMBL474050 0.74 CYP11B2 (0.40) CYP11B2KCNJ1CTSC
SCHEMBL474017 0.73 KCNJ1 (0.33) CYP11B2KCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108903-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed