SCHEMBL473961

SCHEMBL473961

CC(c1c(C(=O)O)cccc1-c1ccccc1)C(O)(c1ccc2c(c1)oc(=O)n2C)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
MAPT P10636 2/20 0.39
THRB P10828 2/20 0.39
CMA1 P23946 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
CYP11B2 P19099 1/20 0.38
CTSG P08311 1/20 0.37
CYP2C8 P10632 1/20 0.37
CYP2C9 P11712 1/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 2/20 0.37
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.35
ASAH1 Q13510 1/20 0.35
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474057 0.94 KMO (0.36) ALDH1A1HPGDMAPTTHRBCMA1
SCHEMBL474521 0.86 TP53 (0.39) ALDH1A1CMA1SMN1; SMN2
SCHEMBL473904 0.82 ALDH1A1 (0.46) ALDH1A1HPGDMAPTTHRBSMN1; SMN2
SCHEMBL473903 0.78 ALDH1A1 (0.37) ALDH1A1MAPTTHRBCMA1CYP11B2
SCHEMBL474051 0.76 ALDH1A1 (0.39) ALDH1A1HPGDMAPTTHRBKMT2A
SCHEMBL12164118 0.76 CYP11B2 (0.41) ALDH1A1HPGDMAPTTHRBCMA1
SCHEMBL473809 0.76 CYP11B2 (0.41) ALDH1A1HPGDMAPTTHRBCMA1
SCHEMBL473967 0.76 ALDH1A1 (0.41) ALDH1A1HPGDMAPTTHRBSMN1; SMN2
SCHEMBL12164188 0.76 ALDH1A1 (0.41) ALDH1A1HPGDMAPTTHRBSMN1; SMN2
SCHEMBL473871 0.74 CYP11B2 (0.39) ALDH1A1HPGDMAPTTHRBCMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed