SCHEMBL4741182

SCHEMBL4741182

Cc1nc(C(=O)O)c(-c2ccc(C(F)(F)F)cc2)o1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.45
MAPT P10636 1/20 0.43
PPARD Q03181 2/20 0.43
PIN1 Q13526 1/20 0.41
PTPN1 P18031 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
DHODH Q02127 1/20 0.41
PPARG P37231 1/20 0.40
HCRTR1 O43613 2/20 0.40
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
SRD5A2 P31213 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1167244 0.83 PIN1 (0.58) PIN1
SCHEMBL1398803 0.83 PTGS2 (0.50) HCRTR1
SCHEMBL1166974 0.83 IKBKB (0.44) IKBKBMAPT
SCHEMBL4742519 0.82 MAPT (0.52) MAPTDHODH
SCHEMBL15507084 0.81 RAB9A (0.44) SRD5A2
SCHEMBL1167223 0.81 MAPK13 (0.50) MAPTPIN1PTPN1HCRTR1
SCHEMBL19256168 0.80 HSD17B10 (0.40) MAPTPIN1PTPN1HCRTR1
SCHEMBL1167143 0.80 NPC1 (0.45) IKBKB
SCHEMBL8192595 0.78 LMNA (0.43) MAPTPTPN1TRPV1
SCHEMBL7695161 0.78 IKBKB (0.50) IKBKBMAPTPPARDPTPN1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087611-A2 PYRROLIDINE- AND PIPERIDINE- BIS-AMIDE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-07-24 WO disclosed