SCHEMBL4742520

SCHEMBL4742520

CC(C)(C)OC(=O)C1(C(=O)O)CCC1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
FFAR3 O14843 1/20 0.31
BTK Q06187 1/20 0.31
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4829842 0.96 NPSR1 (0.31) CYP4F2CYP4A11FFAR3BTKDGAT1
SCHEMBL23293553 0.94 CYP2C19 (0.32) CYP4F2CYP4A11FFAR3BTK
SCHEMBL7884001 0.92 CYP2C19 (0.31) CYP4F2CYP4A11
SCHEMBL8880684 0.91 RBP4 (0.33) CYP4F2CYP4A11FFAR3DGAT1
Ammonia Solution, Strong SCHEMBL28588874 0.89 RBP4 (0.33) CYP4F2CYP4A11FFAR3DGAT1
SCHEMBL22927448 0.89 DGAT1 (0.33) CYP4F2CYP4A11BTKDGAT1
SCHEMBL30683839 0.85 NPSR1 (0.34) CYP4F2CYP4A11BTKDGAT1
SCHEMBL2146137 0.84 OPRM1 (0.34) CYP4F2CYP4A11
SCHEMBL6355124 0.83 NPSR1 (0.33) CYP4F2CYP4A11DGAT1
SCHEMBL5360795 0.82 USP2 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3972649-B1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS AG (CH) 2026-05-13 EP disclosed
EP-4153242-B1 PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES SERVIER LAB (FR) 2024-05-15 EP disclosed
US-20240042051-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE LES LABORATOIRES SERVIER (FR) 2024-02-08 US disclosed
CN-117136076-A MCL-1 inhibitor antibody drug conjugates and methods of use 诺华股份有限公司 2023-11-28 CN disclosed
EP-4251208-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE Novartis AG (CH) 2023-10-04 EP disclosed
US-20230218778-A1 PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES LES LABORATOIRES SERVIER (FR) 2023-07-13 US disclosed
CN-116137818-A Para-amino-benzyl linkers, methods of making and use thereof in conjugates 法国施维雅药厂 2023-05-19 CN disclosed
EP-4153242-A1 PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES Les Laboratoires Servier (FR) 2023-03-29 EP disclosed
US-20230092679-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2023-03-23 US disclosed
US-20230081720-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2023-03-16 US disclosed
US-10124069-B2 Peptidomimetic compounds and antibody-drug conjugates thereof GENENTECH, INC. (US) 2018-11-13 US disclosed
EP-3307780-A1 ANTIBODIES AND IMMUNOCONJUGATES Genentech, Inc. (US) 2018-04-18 EP disclosed
CN-107106700-A Peptide simulated compound and its antibody drug conjugate 基因泰克公司 2017-08-29 CN disclosed
WO-2016205176-A1 ANTIBODIES AND IMMUNOCONJUGATES GENENTECH, INC. (US) 2016-12-22 WO disclosed
EP-3082875-A2 PEPTIDOMIMETIC COMPOUNDS AND ANTIBODY-DRUG CONJUGATES THEREOF Genentech, Inc. (US) 2016-10-26 EP disclosed
US-20160279261-A1 PEPTIDOMIMETIC COMPOUNDS AND ANTIBODY-DRUG CONJUGATES THEREOF GENENTECH, INC. (US) 2016-09-29 US disclosed
WO-2015095227-A2 PEPTIDOMIMETIC COMPOUNDS AND ANTIBODY-DRUG CONJUGATES THEREOF GENENTECH, INC. (US) 2015-06-25 WO disclosed
US-20080207528-A1 Administering derivatives of 4-(3-pyrrolidinyloxy)quinoline TAIGEN BIOTECHNOLOGY CO., LTD. (TW) 2008-08-28 US disclosed
WO-2008095058-A1 HCV PROTEASE INHIBITORS TAIGEN BIOTECHNOLOGY CO. LTD. (TW) 2008-08-07 WO disclosed
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230092679-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE MCL1, BCL9, BAK1 CYP4F2 4666/4885CYP4A11 4779/4885FFAR3 4823/4885
US-20080207528-A1 Administering derivatives of 4-(3-pyrrolidinyloxy)quinoline GLS2, SLC10A1, UGT1A1 CYP4F2 8/4885CYP4A11 58/4885FFAR3 3170/4885
US-20230081720-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE MCL1, CD74, CD99 CYP4F2 3887/4885CYP4A11 4814/4885FFAR3 4752/4885
US-20240042051-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE MCL1, CD58, LENG8 CYP4F2 4168/4885CYP4A11 4847/4885FFAR3 4774/4885
US-20230218778-A1 PARA-AMINO-BENZYL LINKERS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN CONJUGATES DNPEP, PEPD, PREP CYP4F2 421/4885CYP4A11 1045/4885FFAR3 3981/4885
US-20160279261-A1 PEPTIDOMIMETIC COMPOUNDS AND ANTIBODY-DRUG CONJUGATES THEREOF DNPEP, LNPEP, BCR CYP4F2 3842/4885CYP4A11 4396/4885FFAR3 2922/4885
US-10124069-B2 Peptidomimetic compounds and antibody-drug conjugates thereof DNPEP, LNPEP, BCR CYP4F2 3842/4885CYP4A11 4396/4885FFAR3 2922/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.