SCHEMBL4742574

SCHEMBL4742574

COCCN1CCN(c2c(C(=O)NC(CC(=O)OC(=O)C(F)(F)F)C(=O)CF)cnc3c([N+](=O)[O-])cccc23)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.35
DRD3 P35462 3/20 0.35
MAPT P10636 5/20 0.34
MAPK1 P28482 4/20 0.34
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.34
PKM P14618 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
USP2 O75604 1/20 0.33
TP53 P04637 1/20 0.33
RECQL P46063 1/20 0.33
HSD17B10 Q99714 1/20 0.33
LMNA P02545 3/20 0.32
NPSR1 Q6W5P4 2/20 0.32
HTT P42858 2/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742160 0.92 MEN1 (0.36) DRD2DRD3MAPTMAPK1ALDH1A1
SCHEMBL4739351 0.92 MAPK1 (0.35) MAPTMAPK1ALDH1A1KDM4EPKM
Trifluoroacetic Acid SCHEMBL4742566 0.90 DRD2 (0.35) DRD2DRD3MAPTMAPK1ALDH1A1
SCHEMBL4742618 0.88 USP2 (0.34) MAPTMAPK1USP2TP53RECQL
Trifluoroacetic Acid SCHEMBL4742157 0.82 MEN1 (0.36) MAPTMAPK1ALDH1A1KDM4EPKM
Trifluoroacetic Acid SCHEMBL4739344 0.82 SIRT6 (0.36) MAPTMAPK1ALDH1A1USP2TP53
SCHEMBL4743406 0.80 MET (0.39) MAPTMAPK1ALDH1A1KDM4EUSP2
SCHEMBL4743039 0.78 USP2 (0.35) MAPTMAPK1ALDH1A1KDM4EUSP2
SCHEMBL4739980 0.70 THRB (0.44) MAPTALDH1A1SMN1; SMN2
SCHEMBL4742621 0.70 USP2 (0.45) MAPTMAPK1KDM4EUSP2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed